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Christopher S Burgey Selected Research

Calcitonin Gene-Related Peptide Receptor Antagonists

1/2020Characterization of Ubrogepant: A Potent and Selective Antagonist of the Human Calcitonin Gene‒Related Peptide Receptor.
11/2015Novel oxazolidinone calcitonin gene-related peptide (CGRP) receptor antagonists for the acute treatment of migraine.
5/2011Orally bioavailable imidazoazepanes as calcitonin gene-related peptide (CGRP) receptor antagonists: discovery of MK-2918.
1/2009Examining the binding properties of MK-0974: a CGRP receptor antagonist for the acute treatment of migraine.
1/2009Calcitonin gene-related peptide receptor antagonists for the treatment of migraine.
8/2008Synthesis of the (3R,6S)-3-amino-6-(2,3-difluorophenyl)azepan-2-one of telcagepant (MK-0974), a calcitonin gene-related peptide receptor antagonist for the treatment of migraine headache.
2/2008Pharmacological characterization of MK-0974 [N-[(3R,6S)-6-(2,3-difluorophenyl)-2-oxo-1-(2,2,2-trifluoroethyl)azepan-3-yl]-4-(2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl)piperidine-1-carboxamide], a potent and orally active calcitonin gene-related peptide receptor antagonist for the treatment of migraine.
1/2008Calcitonin gene-related peptide (CGRP) receptor antagonists: investigations of a pyridinone template.
11/2007Potent, orally bioavailable calcitonin gene-related peptide receptor antagonists for the treatment of migraine: discovery of N-[(3R,6S)-6-(2,3-difluorophenyl)-2-oxo-1- (2,2,2-trifluoroethyl)azepan-3-yl]-4- (2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin- 1-yl)piperidine-1-carboxamide (MK-0974).
9/2007Caprolactams as potent CGRP receptor antagonists for the treatment of migraine.
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Christopher S Burgey Research Topics

Disease

11Migraine Disorders (Migraine)
01/2020 - 10/2006
2Pain (Aches)
01/2022 - 06/2021
1Postoperative Pain
01/2021
1Neuroblastoma
01/2009

Drug/Important Bio-Agent (IBA)

11Calcitonin Gene-Related Peptide Receptor AntagonistsIBA
01/2020 - 10/2006
6Calcitonin Gene-Related PeptideIBA
01/2020 - 09/2007
3telcagepantIBA
01/2009 - 02/2008
2Calcitonin Gene-Related Peptide Receptors (Calcitonin-Gene Related Peptide Receptor)IBA
01/2020 - 01/2009
2NeuropeptidesIBA
01/2009 - 02/2008
2piperidineIBA
02/2008 - 11/2007
1Peptides (Polypeptides)IBA
01/2022
1Voltage-Gated Sodium ChannelsIBA
06/2021
1Protein Isoforms (Isoforms)IBA
06/2021
1Analgesics (Analgesic Drugs)IBA
01/2021
1ubrogepantIBA
01/2020
1Monoclonal AntibodiesIBA
01/2020
1Oxazolidinones (2 Oxazolidone)IBA
11/2015
1olcegepantIBA
02/2008
1PiperidinesIBA
10/2006
1BenzodiazepinesIBA
10/2006

Therapy/Procedure

2Therapeutics
06/2021 - 02/2008